溶解性 | DMSO 100 mg/mL Water 100 mg/mL Ethanol <1 mg/mL |
存贮条件 | 储存温度-20°C |
备注 | GZD824 is a novel orally bioavailable Bcr-Abl inhibitor for Bcr-Abl(WT) and Bcr-Abl(T315I) with IC50 of 0.34 nM and 0.68 nM, respectively. |
别名 | Benzamide, 4-methyl-N-[4-[(4-methyl-1-piperazinyl)methyl]-3-(trifluoromethyl)phenyl]-3-[2-(1H-pyrazolo[3,4-b]pyridin-5-yl)ethynyl]-, methanesulfonate (1:2);Benzamide, 4-methyl-N-[4-[(4-methyl-1-piperazinyl)methyl]-3-(trifluoromethyl)phenyl]-3-[2-(1H-pyrazolo[3,4-b]pyridin-5-yl)ethynyl]-, methanesulfonate (1:2) |
GZD824,Bcr-Abl抑制剂
GZD824 Dimesylate (订货以英文为准)
编号:G129296
CAS号:1421783-64-3
分子式:C31H35F3N6O7S2
分子量:724.77
产品名称 | GZD824 Dimesylate |
中文名称 | GZD824,Bcr-Abl抑制剂 |
CAS号 | 1421783-64-3 |
分子式(M.F.) | C31H35F3N6O7S2 |
分子量(M.W.) | 724.77 |
储存条件 | 避光;-20°C储存 |
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